Reuptake inhibitor
A reuptake inhibitor (RI), also known as a transporter blocker, is a drug that inhibits the plasmalemmal transporter-mediated reuptake of a neurotransmitter from the synapse into the pre-synaptic neuron, leading to an increase in the extracellular concentrations of the neurotransmitter and therefore an increase in neurotransmission.
Reuptake inhibitorSerotonin reuptake inhibitorNorepinephrine reuptake inhibitorDopamine reuptake inhibitorSelective serotonin reuptake inhibitorMonoamine reuptake inhibitorGABA reuptake inhibitorSerotonin-dopamine reuptake inhibitorAllosteric serotonin reuptake inhibitorSerotonin–norepinephrine reuptake inhibitorSerotonin–norepinephrine–dopamine reuptake inhibitorNorepinephrine-dopamine reuptake inhibitorAdenosine reuptake inhibitorAntidepressantSSRI discontinuation syndromeEndocannabinoid reuptake inhibitorDiscovery and development of dual serotonin and norepinephrine reuptake inhibitorsSertralineSerotoninFluoxetine




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